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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T60849 | PIN1 inhibitor 2 | ||
PIN1 inhibitor 2 (compound 12) is a potent inhibitor of PIN1 that has the potential in the breast cancer research. PIN1 inhibitor 2 exhibits antitumor activity with an IC 50 of 9.55 μM against MCF7 cells [1]. | |||
T9240 | Sulfopin | Acetamide, 2-chloro-N-(2,2-dimethylpropyl)-N-(tetrahydro-1,1-dioxido-3-thienyl)- | Others |
Sulfopin is a highly selective covalent inhibitor of Pin1 with an apparent Ki of 17nM. Sulfopin blocks Myc-driven tumors in vivo. |